Dr. Athanasios Markos
Research Interests
Development of new bioorthogonal reactions
Curriculum Vitae
Publications
A. Markos, M. Biedermann, J. Heimgärtner, A. Schmitt, K. Lang, H. Wennemers "Introducing Azomethine Imines to Chemical Biology: Bioorthogonal Reaction with Isonitriles"
J. Am. Chem. Soc. 2023, 145, 19513-19517.
A. Markos, L. Janecky, B. Klepetarova, R. Pohl and P. Beier “Stereoselective Synthesis of (Z)-β-Enamido Fluorides from N-Fluoroalkyl- and N-Sulfonyl-1,2,3-Triazoles”
Org. Lett. 2021, 23, 4224.
A. Markos, L. Janecky, T. Chvojka, T. Martinek, H. Martines-Seara, B. Klepetarova, and P. Beier “Haloalkenyl Imidoyl Halides as Multifacial Substrates in the Stereoselective Synthesis of N-Alkenyl Compounds”
Adv. Synth. Catal. 2021, 363, 3258.
V. Motornov, V. Kostal, A. Markos, D. Täffner and P. Beier “General Approach to 2-Fluoroalkyl 1,3-Azoles via the Tandem Ring Opening and Defluorinative Annulation of N-Fluoroalkyl-1,2,3-Triazoles”
Org. Chem. Front. 2019, 6, 3776.
A. Markos, S. Voltrova, V. Motornov, D. Tichy, B. Klepetarova and Beier, P. “Stereoselective Synthesis of (Z)-β-Enamido Triflates and Fluorosulfonates from N-Fluoroalkylated Triazoles”
Chem. Eur. J. 2019, 25, 7640.
V. Motornov, A. Markos and P. Beier A “Rhodium-Catalyzed Transannulation of N-(per)Fluoroalkyl-1,2,3-Triazoles under Microwave Conditions - a General Route to N-(per)Fluoroalkyl-Substituted Five-Membered Heterocycles”
Chem. Commun. 2018, 54, 3258.
K. Burglova, G. Rylova, A. Markos, H. Prichystalova, M. Soural, M. Petracek, M. Medvedikova, G. Tejral, B. Sopko, P. Hradil, P, Dzubak, M. Hajduch and J. Hlavac. “Identification of Eukaryotic Translation Elongation Factor 1-α1 Gamendazole-Binding Site for Binding of 3-Hydroxy-4(1H)-Quinolinones as Novel Ligands with Anticancer Activity”
J. Med. Chem. 2018, 61, 3027.